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Found 1 Enz. Inhib. hit(s) with Target = 'ATP-dependent translocase ABCB1' and Ligand = 'BDBM50119426'
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50119426(30-Ethyl-6,9,18,24,33-pentaisobutyl-3,21-diisoprop...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity against Human MDR1 P-Glycoprotein ABC Transporter using leukemia CEM cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed