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Found 3 Enz. Inhib. hit(s) with Target = 'Acetylcholinesterase' and Ligand = 'BDBM192119'
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192119(2-(4-(1-(2,4-dinitrobenzoyl)-3-(1H-indol-3-yl)-4,5...)
Affinity DataIC50:  1.60E+4nMT: 2°CAssay Description:Preparation of DPPH solution was adopted from Molyneux [J. Sci. Technol. 26(2):211-219] and Blois [Nature 181(4617):1199-1200] with minor modificatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192119(2-(4-(1-(2,4-dinitrobenzoyl)-3-(1H-indol-3-yl)-4,5...)
Affinity DataIC50:  1.62E+4nMT: 2°CAssay Description:The ABTS free radical cation scavenging ability of the synthe- sized compounds was determined according to the procedure described earlier [Free Radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Aimst University

LigandPNGBDBM192119(2-(4-(1-(2,4-dinitrobenzoyl)-3-(1H-indol-3-yl)-4,5...)
Affinity DataIC50:  2.71E+4nMpH: 8.0 T: 2°CAssay Description:The in vitro AChE inhibitory activity was measured using the methods described earlier [Biochem. Pharmacol. 7:88-95]. Briefly, stock solutions (1mg/m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed