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Found 2 Enz. Inhib. hit(s) with Target = 'Acetylcholinesterase' and Ligand = 'BDBM29402'
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Csic

LigandPNGBDBM29402(tacrine-dihydropyridine hybrid (tacripyrine), 13)
Affinity DataIC50:  47nMAssay Description:The inhibitory activity of the compounds towards AChE was determined following the spectrophotometric method of Rappaport using purified AChE from Ee...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Csic

LigandPNGBDBM29402(tacrine-dihydropyridine hybrid (tacripyrine), 13)
Affinity DataIC50:  158nMpH: 7.2 T: 2°CAssay Description:The inhibitory activity of the compounds towards hAChE was determined following the method of Ellman using AChE from human serum and acetylthiocholin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed