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Found 5 Enz. Inhib. hit(s) with Target = 'Acetylcholinesterase' and Ligand = 'BDBM50244216'
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50244216(2,3-dihydropyrrolo[2,1-b]quinazolin-9(1H)-one | CH...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50244216(2,3-dihydropyrrolo[2,1-b]quinazolin-9(1H)-one | CH...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of Electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by addition of substrate and measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Louisiana At Lafayette

Curated by ChEMBL
LigandPNGBDBM50244216(2,3-dihydropyrrolo[2,1-b]quinazolin-9(1H)-one | CH...)
Affinity DataIC50:  3.52E+4nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Louisiana At Lafayette

Curated by ChEMBL
LigandPNGBDBM50244216(2,3-dihydropyrrolo[2,1-b]quinazolin-9(1H)-one | CH...)
Affinity DataIC50:  6.25E+4nMAssay Description:Inhibition of human AChE pre-incubated for 6 mins before ATCI substrate addition and measured after 12 mins by DTNB reagent dependent UV-Vis spectrop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Louisiana At Lafayette

Curated by ChEMBL
LigandPNGBDBM50244216(2,3-dihydropyrrolo[2,1-b]quinazolin-9(1H)-one | CH...)
Affinity DataIC50:  8.25E+4nMAssay Description:Inhibition of AchE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed