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Found 2 Enz. Inhib. hit(s) with Target = 'Acyl-CoA:cholesterol acyltransferase' and Ligand = 'BDBM50065002'
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50065002(1-(4-Dimethylamino-benzyl)-3-(6-methyl-2,4-bis-met...)
Affinity DataIC50:  72nMAssay Description:In vitro inhibitory activity against Acyl coenzyme A:cholesterol acyltransferase (ACAT) in rabbit intestinal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50065002(1-(4-Dimethylamino-benzyl)-3-(6-methyl-2,4-bis-met...)
Affinity DataIC50:  72nMAssay Description:In vitro inhibitory activity towards ACAT by the displacement of [1-14C]-oleolyl-CoA from the small intestine of cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed