Found 34 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM35804' 
Affinity DataKi: 289nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 289nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 289nMAssay Description:Binding affinity for human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Agonist activity at human adenosine receptor A1More data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Binding affinity to human recombinant adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 302nMAssay Description:Inhibition of [3H]DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 380nMAssay Description:Displacement of [3H]R-PIA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 380nMAssay Description:Displacement of [3H]N6-phenylisopropyladenosine from human A1 adenosine receptor expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 569nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 569nMAssay Description:Binding affinity against adenosine A1 receptor from rat brain using [3H]CHA as a radioligand.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 1.14E+3nMAssay Description:Binding affinity against adenosine A1 receptor from rat brain membranes using [3H]cyclohexyladenosine as radioligand.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 1.23E+3nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]CHA as radioligandMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 1.23E+3nMAssay Description:Inhibition of [3H]CHA binding to adenosine A1 receptor from rat brain membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 1.41E+3nMAssay Description:Adenosine A1 receptor binding was measured in adenosine deaminase (ADA) pretreated rat cortical membranes using [3H]cyclohexyladenosine in the presen...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 1.80E+3nMAssay Description:Binding affinity towards adenosine A1 receptor in rat brain cortexMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 1.80E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 1.80E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortexMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 2.60E+3nMAssay Description:Inhibition of [3H]PIA binding to rat cortical adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 2.60E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]-CHA or [3H]PIA as radioligandMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 2.60E+3nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in rat cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 2.60E+3nMAssay Description:Displacement of [3H]- DPCPX from adenosine A1 receptor on rat cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 2.60E+3nMAssay Description:Tested for the binding affinity of A1 receptor by displacing the [3H]-PIA in rat brain membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 9.90E+3nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of Wistar rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cell membranes incubated for 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataEC50: 2.46E+4nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human adenosine A1 receptor expressed in CHO cells by GTPPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.44E+3nMAssay Description:Binding against human adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataEC50: >100nMAssay Description:[S]GTP gamma-S binding against adenosine A1 receptor in rat brainMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
Affinity DataEC50: 6.31E+5nMAssay Description:Agonist activity at human Adenosine A1 receptor expressed in yeast cells coexpressed with chimeric GPA1/Galphai1 after 16 hrs by beta galactosidase r...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Zeneca Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataEC50: >1.00E+4nMAssay Description:Activitty at Adenosine A1 receptor of rat atriaMore data for this Ligand-Target Pair
