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Found 5 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50001500'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50001500(7-Methyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione...)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of 1 nM [3H]- N6-(phenylisopropyl) adenosine binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50001500(7-Methyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione...)
Affinity DataKi:  7.00E+3nMAssay Description:Binding affinity to A1 adenosine receptor from rat cortical membrane in presence of [3H]-R-(phenylisopropyl)-adenosineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50001500(7-Methyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione...)
Affinity DataKi:  7.00E+3nMAssay Description:Ability to inhibit binding of 1 nM [3H]-cyclohexyladenosine to adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50001500(7-Methyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione...)
Affinity DataKi:  7.70E+3nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50001500(7-Methyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione...)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibition of 1 nM [3H]- N6 -(phenylisopropyl) adenosine binding to Adenosine A1 receptor in rat fat cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed