Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50088423'
TargetAdenosine receptor A1(Rat)
Niddk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50088423BDBM50088423((1R,2R,3S,4R,5S)-4-(2-Chloro-6-cyclopentylamino-pu...)
Affinity DataKi:  8.80nMAssay Description:Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Niddk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50088423BDBM50088423((1R,2R,3S,4R,5S)-4-(2-Chloro-6-cyclopentylamino-pu...)
Affinity DataKi:  8.80nMAssay Description:Displacement of [3H]R-PIA from rat brain membrane Adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50088423BDBM50088423((1R,2R,3S,4R,5S)-4-(2-Chloro-6-cyclopentylamino-pu...)
Affinity DataEC50:  31nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding to human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Niddk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50088423BDBM50088423((1R,2R,3S,4R,5S)-4-(2-Chloro-6-cyclopentylamino-pu...)
Affinity DataEC50:  145nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding to adenosine A1 receptor of rat cerebral cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed