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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50452336'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50452336(CHEMBL2113406)
Affinity DataKi:  7.5nMAssay Description:Affinity for adenosine A1 receptor at rat cortical receptors using 1 nM [3H]PIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50452336(CHEMBL2113406)
Affinity DataKi:  16nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50452336(CHEMBL2113406)
Affinity DataKi:  864nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membrane incubated for 60 mins by microplate beta scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed