Affinity DataKi: 4nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 475nMAssay Description:Negative chronotropic activity for A1 Adenosine receptor in spontaneously beating rat atriaMore data for this Ligand-Target Pair