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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a/A2b' and Ligand = 'BDBM50018157'
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50018157(1-Methyl-8-phenyl-3,7-dihydro-purine-2,6-dione | C...)
Affinity DataKi:  250nMAssay Description:Inhibition of the stimulation by 5'-(N-ethylcarbamoyl) adenosine of adenyl cyclase via Adenosine A2 receptor in rat PC12 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50018157(1-Methyl-8-phenyl-3,7-dihydro-purine-2,6-dione | C...)
Affinity DataKi:  860nMAssay Description:Inhibition of 1 nM [3H]- N6 -(phenylisopropyl) adenosine binding to Adenosine A1 receptor in rat fat cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50018157(1-Methyl-8-phenyl-3,7-dihydro-purine-2,6-dione | C...)
Affinity DataKi:  2.20E+3nMAssay Description:Binding affinity against Adenosine A2 receptor in rat striatal membranes using [3H]5'-(N-ethylcarboxamido)-adenosine (NECA) as the ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed