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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a/A2b' and Ligand = 'BDBM50453222'
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50453222(CHEMBL2113509)
Affinity DataKi:  13nMAssay Description:Inhibition of adenylate cyclase via A1 receptors in rat fat cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50453222(CHEMBL2113509)
Affinity DataKi:  20nMAssay Description:Binding affinity against high affinity component of adenosine A1 receptors from rat brain membranes using [3H]DPCPXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50453222(CHEMBL2113509)
Affinity DataEC50:  62nMAssay Description:Binding affinity against Adenosine A2 receptor from rat striatal membranes with 50 nM CPA using [3H]-NECAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed