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Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a/A2b' and Ligand = 'BDBM50453223'
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
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Curated by ChEMBL
LigandPNGBDBM50453223(CHEMBL2113507)
Affinity DataKi:  2.80nMAssay Description:Inhibition of adenylate cyclase via adenosine A1 receptors in rat fat cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
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Curated by ChEMBL
LigandPNGBDBM50453223(CHEMBL2113507)
Affinity DataKi:  5.40nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatal membranes using [3H]NECA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50453223(CHEMBL2113507)
Affinity DataKi:  21nMAssay Description:Binding affinity against adenosine A2 receptor from human platelet membranes using [3H]NECAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50453223(CHEMBL2113507)
Affinity DataEC50:  414nMAssay Description:Maximal NECA stimulation of adenylate cyclase via adenosine A2 receptor in human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed