Affinity DataKi: 3.80nMAssay Description:Binding affinity against adenosine A2 receptor from rat striatal membranes with 50 nM CPA using [3H]-NECAMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Binding affinity against adenosine A2 receptor from rat striatum using [3H]NECA as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Binding affinity against adenosine A2 receptor from human platelet membranes using [3H]NECAMore data for this Ligand-Target Pair
Affinity DataEC50: 105nMAssay Description:Inhibition of adenylate cyclase via Adenosine A1 receptor in rat fat cell membranesMore data for this Ligand-Target Pair