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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50061931'
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Julius-Maximilians-UniversitäT WüRzburg

Curated by ChEMBL
LigandPNGBDBM50061931(8-[(E)-2-(3-Chloro-phenyl)-vinyl]-3,7-dimethyl-1-p...)
Affinity DataKi:  13nMAssay Description:Ability to inhibit binding of [3H]-CGS- 21680 to adenosine A2A receptor in rat brain striatal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Julius-Maximilians-UniversitäT WüRzburg

Curated by ChEMBL
LigandPNGBDBM50061931(8-[(E)-2-(3-Chloro-phenyl)-vinyl]-3,7-dimethyl-1-p...)
Affinity DataKi:  47nMAssay Description:Ability to inhibit binding of [3H]-NECA to Adenosine A2A receptor in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed