Affinity DataKi: 3.60nMAssay Description:Binding affinity to human adenosine A2A receptor measured by radioligand-based affinity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.00190nMAssay Description:Inverse agonist activity at human adenosine A2A receptor expressed in CHO cells assessed as inhibition of cAMP accumulation measured after 150 mins i...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0510nMAssay Description:Antagonist activity against human adenosine A2A receptor expressed in CHO cells assessed as inhibition of CGS21680-stimulated cAMP accumulation measu...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inverse agonist activity at human A2A receptor assessed as inhibition of cAMP accumulationMore data for this Ligand-Target Pair