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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50275803'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50275803(CHEMBL469324 | N-(2-(3,5-dimethyl-1H-pyrazol-1-yl)...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50275803(CHEMBL469324 | N-(2-(3,5-dimethyl-1H-pyrazol-1-yl)...)
Affinity DataIC50:  42nMAssay Description:Activity at adenosine A2A receptor in rat PC12 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed