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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50318244'
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50318244((R)-N-(3-phenyl-1H-1,2,4-triazol-5-yl)-2-(m-tolylo...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]CGS21680 from human recombinant adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50318244((R)-N-(3-phenyl-1H-1,2,4-triazol-5-yl)-2-(m-tolylo...)
Affinity DataKi:  200nMAssay Description:Displacement of radioligand from human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50318244((R)-N-(3-phenyl-1H-1,2,4-triazol-5-yl)-2-(m-tolylo...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]CGS21680 from human A2A adenosine receptor expressed in HEK293 cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed