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Found 6 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50364045'
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50364045(CHEMBL1950554)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in rat brain striatal membrane after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50364045(CHEMBL1950554)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]CGS21680 from human recombinant adenosine A2A receptor expressed in HEK cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50364045(CHEMBL1950554)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]CGS21680 from human recombinant adenosine A2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50364045(CHEMBL1950554)
Affinity DataKi:  270nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50364045(CHEMBL1950554)
Affinity DataKi:  270nMAssay Description:Binding affinity to human recombinant adenosine receptor A2aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50364045(CHEMBL1950554)
Affinity DataKi:  270nMAssay Description:Binding affinity to A2A adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed