Affinity DataKi: 24nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity to human adenosine A2B receptor at 10 uMMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of human A2B adenosine receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in HEK293 cells assessed as inhibition of NECA-induced increase of intracellular cAMP l...More data for this Ligand-Target Pair
Affinity DataIC50: 512nMAssay Description:Antagonist activity at mouse adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-induced increase of intracellular cAMP leve...More data for this Ligand-Target Pair