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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50086147'
TargetAdenosine receptor A3(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50086147(4-Amino-2-m-tolyl-2H-[1,2,4]triazolo[4,3-a]quinoxa...)
Affinity DataKi:  28.5nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50086147(4-Amino-2-m-tolyl-2H-[1,2,4]triazolo[4,3-a]quinoxa...)
Affinity DataKi:  28.5nMAssay Description:Binding affinity towards human adenosine A3 receptor expressed in HEK-293 cells in presence of [125I]-AB-MECA at a concentration of 1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed