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Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50158776'
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50158776(1-(2-Furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2...)
Affinity DataKi:  9nMAssay Description:Binding affinity for human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50158776(1-(2-Furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2...)
Affinity DataKi:  9nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50158776(1-(2-Furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2...)
Affinity DataKi:  9nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50158776(1-(2-Furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2...)
Affinity DataKi:  8.91E+3nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed