Affinity DataKi: 32nMAssay Description:Displacement of [125I]I-AB-MECA from human recombinant adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in CHO cells assessed as blockade of Cl-IB-MECA-mediated inhibition of forskolin-stimula...More data for this Ligand-Target Pair
Affinity DataKd: 0.158nMAssay Description:Antagonist activity at human recombinant adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair