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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50573587'
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573587(CHEMBL4861092)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in HeLa cell membrane incubated for 180 mins by microplate beta scintillation cou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573587(CHEMBL4861092)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human adenosine A3 receptor transfected in CHO cells assessed as cAMP level measured after 35 mins by cAMP enzyme immunoassayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed