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Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50602677'
TargetAdenosine receptor A3(Mus musculus)
National Institute Of Diabetes And Digestive And Kidney Disease

Curated by ChEMBL
LigandPNGBDBM50602677(CHEMBL5170037)
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I] N6-4-amino-3-iodobenzyl adenosine 5-N-methyluronamide from mouse A3A receptor stably expressed in HEK293 cell membrane by radi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Disease

Curated by ChEMBL
LigandPNGBDBM50602677(CHEMBL5170037)
Affinity DataKi:  3.30nMAssay Description:Displacement of [125I] N6-(4-amino-3-iodobenzyl)adenosine-5'-N-methyluronamide from human A3A receptor stably expressed in HEK293 cell membrane by ra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Disease

Curated by ChEMBL
LigandPNGBDBM50602677(CHEMBL5170037)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human adenosine A3A receptor stably expressed in HEK293 cells assessed as mini G-alpha recruitment potency by luciferase based Na...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Disease

Curated by ChEMBL
LigandPNGBDBM50602677(CHEMBL5170037)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human adenosine A3A receptor stably expressed in HEK293 cells assessed as beta arrestin 2 recruitment potency by luciferase based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed