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Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-1A adrenergic receptor' and Ligand = 'BDBM50238834'
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238834(2-(5-chloro-4-(1H-pyrazol-4-yl)-2,3-dihydro-1H-ind...)
Affinity DataEC50:  78nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238834(2-(5-chloro-4-(1H-pyrazol-4-yl)-2,3-dihydro-1H-ind...)
Affinity DataEC50:  78nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells by calcium mobilization-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed