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Found 3 Enz. Inhib. hit(s) with Target = 'Alpha-1A adrenergic receptor' and Ligand = 'BDBM50392645'
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50392645(CHEMBL2153557)
Affinity DataKi:  0.646nMAssay Description:Displacement of [3H]prazosin from human cloned alpha1A adrenoceptor expressed in CHO cell membranes after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
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Curated by ChEMBL
LigandPNGBDBM50392645(CHEMBL2153557)
Affinity DataKd:  28.8nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat prostatic vas deferans assessed as inhibition of noradrenaline-induced contractions...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50392645(CHEMBL2153557)
Affinity DataKd:  1.20nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat prostate assessed as inhibition of noradrenaline-induced contractions after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed