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Found 3 Enz. Inhib. hit(s) with Target = 'Alpha-1A adrenergic receptor' and Ligand = 'BDBM50474671'
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474671(CHEMBL111554)
Affinity DataKi:  195nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474671(CHEMBL111554)
Affinity DataKi:  195nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50474671(CHEMBL111554)
Affinity DataEC50:  447nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article