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Found 3 Enz. Inhib. hit(s) with Target = 'Alpha-1B adrenergic receptor' and Ligand = 'BDBM50274049'
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50274049(CHEMBL342062)
Affinity DataKi:  0.0708nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50274049(CHEMBL342062)
Affinity DataKi:  0.135nMAssay Description:Compound was tested for binding affinity against human hippocampus Alpha-1B adrenergic receptor using radioligand ([3H]-prazosin) binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50274049(CHEMBL342062)
Affinity DataKi:  0.692nMAssay Description:Compound was tested for binding affinity against cloned Alpha-1B adrenergic receptor from hamster smooth muscle using radioligand ([3H]prazosin) bind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed