Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Alpha-1B adrenergic receptor' and Ligand = 'BDBM50487287'
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50487287((+)-CYCLAZOSIN)
Affinity DataKi:  0.135nMAssay Description:Displacement of [3H]prazosin from Homo sapiens (human) alpha1B adrenergic receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50487287((+)-CYCLAZOSIN)
Affinity DataKi:  0.209nMAssay Description:Binding affinity to alpha1B adrenoreceptor in Rattus norvegicus (rat) liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50487287((+)-CYCLAZOSIN)
Affinity DataKi:  0.692nMAssay Description:Binding affinity to alpha1B adrenoreceptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article