Affinity DataKi: 0.0380nMAssay Description:Displacement of [3H]prazosin from human recombinant adrenergic alpha-1B receptor expressed in CHO cell membranes incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:The binding affinity was evaluated on cloned human alpha-1B adrenergic receptor expressed in chinese hamster ovary(CHO) cells by using [3H]prazosin a...More data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Overall binding displacement in tissues containing only the Alpha-1B adrenergic receptor (rat spleen, rat liver)More data for this Ligand-Target Pair
Affinity DataKi: 9.90nMAssay Description:Binding affinity against Alpha-1B adrenergic receptor from human cloneMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]prazosin from human recombinant alpha1B adrenergic receptor expressed in CHO cell membranes after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]prazosin from human cloned Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity measured in CHO cells expressing human cloned Alpha-1B adrenergic receptor expressed as pKiMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]prazosin from human cloned Alpha-1B adrenoreceptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]prazosin from human adrenergic Alpha-1B expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 25.6nMAssay Description:Binding affinity of the compound towards Alpha-1B adrenergic receptor native receptor in rat liver using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Binding affinity against Alpha-1B adrenergic receptor from hamster clones.More data for this Ligand-Target Pair
Affinity DataKi: 57.3nMAssay Description:Binding affinity of the compound towards Alpha-1B adrenergic receptor cloned receptor hamster smooth muscle using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair