Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Alpha-1D adrenergic receptor' and Ligand = 'BDBM50118705'
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataKi:  275nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataKi:  275nMAssay Description:In vitro binding affinity towards alpha-1D adrenergic receptor of rat clone in radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataKi:  280nMAssay Description:Binding affinity towards rat cloned Alpha-1D adrenergic receptor ; value ranges from (0.24 -0.32)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed