Affinity DataKi: 91nMAssay Description:Inhibitory constant against human Alpha-2B adrenergic receptor expressed in Y-1 cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataEC50: 562nMAssay Description:Alpha-2B adrenergic receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair