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Found 4 Enz. Inhib. hit(s) with Target = 'Alpha-2C adrenergic receptor' and Ligand = 'BDBM50052880'
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Allergan

Curated by ChEMBL
LigandPNGBDBM50052880(CHEMBL49137 | Imidazolidin-2-ylidene-(5-methyl-qui...)
Affinity DataKi:  27nMAssay Description:Compound was tested in vitro for binding affinity against Alpha-2C adrenergic receptor from cloned human C-2 receptor transfected into Chinese hamste...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Allergan

Curated by ChEMBL
LigandPNGBDBM50052880(CHEMBL49137 | Imidazolidin-2-ylidene-(5-methyl-qui...)
Affinity DataKi:  27nMAssay Description:Displacement of rauwolscine from human Alpha-2C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Allergan

Curated by ChEMBL
LigandPNGBDBM50052880(CHEMBL49137 | Imidazolidin-2-ylidene-(5-methyl-qui...)
Affinity DataKi:  28nMAssay Description:Binding affinity for human Alpha-2C adrenergic receptor from cultured LM(tk-) cells using [3H]- prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Allergan

Curated by ChEMBL
LigandPNGBDBM50052880(CHEMBL49137 | Imidazolidin-2-ylidene-(5-methyl-qui...)
Affinity DataEC50:  14nMAssay Description:Alpha-2C adrenergic receptor agonistic potency as inhibition of forskolin-stimulated cyclic adenosine monophosphate synthesisMore data for this Ligand-Target Pair
In DepthDetails