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Found 4 Enz. Inhib. hit(s) with Target = 'Alpha-2C adrenergic receptor' and Ligand = 'BDBM50417347'
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417347(CHEMBL385310)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417347(CHEMBL385310)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]RX821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417347(CHEMBL385310)
Affinity DataEC50:  93nMAssay Description:Agonist activity at human adrenergic alpha-2C receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417347(CHEMBL385310)
Affinity DataEC50:  93nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed