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Found 6 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] A' and Ligand = 'BDBM50046866'
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50046866(CHEMBL3319256)
Affinity DataIC50:  0.389nMAssay Description:Inhibition of recombinant human MAOA expressed in baculovirus-infected BTI insect cells using p-tyramine as substrate measured for 45 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50046866(CHEMBL3319256)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant MAO-A expressed in baculovirus-infected insect cells using p-tyraimne substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50046866(CHEMBL3319256)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50046866(CHEMBL3319256)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human MAOA expressed in baculovirus-infected BTI insect cells using p-tyramine as substrate measured for 45 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50046866(CHEMBL3319256)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat liver mitochondria using p-tyramine as substrate measured for 45 mins in presence of MAOB inhibitor selegili...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50046866(CHEMBL3319256)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus-infected insect cells using p-tyraimne substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed