Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Amyloid-beta precursor protein' and Ligand = 'BDBM50122785'
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50122785(4-(6-bromoH-imidazo[1,2-a]pyridin-2-yl)-N,N-dimeth...)
Affinity DataKi:  5.90nMAssay Description:Binding affinity to human beta amyloid plaque in alzheimer's disease patient brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50122785(4-(6-bromoH-imidazo[1,2-a]pyridin-2-yl)-N,N-dimeth...)
Affinity DataKi:  10.3nMAssay Description:Inhibition constant against [125I]-7 (TZDM) binding to Amyloid beta 1-40 aggregatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed