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Found 2 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM50063118'
TargetAndrogen receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50063118(3a,10-Dimethyl-7-trifluoromethyl-1,2,3a,4,5,10-hex...)
Affinity DataKi:  78nMAssay Description:Binding affinity for human androgen receptor in transiently-transfected COS-1 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50063118(3a,10-Dimethyl-7-trifluoromethyl-1,2,3a,4,5,10-hex...)
Affinity DataIC50:  27nMAssay Description:Antagonistic activity against human androgen receptor (hAR) in co-transfected CV-1 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed