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Found 2 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM50063124'
TargetAndrogen receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50063124(6,8,8,9-Tetramethyl-4-trifluoromethyl-8,9-dihydro-...)
Affinity DataKi:  695nMAssay Description:Binding affinity for human androgen receptor in transiently-transfected COS-1 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50063124(6,8,8,9-Tetramethyl-4-trifluoromethyl-8,9-dihydro-...)
Affinity DataIC50:  156nMAssay Description:Antagonistic activity against human androgen receptor (hAR) in co-transfected CV-1 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed