Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM50068100'
TargetAndrogen receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50068100(CHEMBL3402231)
Affinity DataIC50:  4.10nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50068100(CHEMBL3402231)
Affinity DataEC50:  1.20nMAssay Description:Modulation of androgen receptor (unknown origin) expressed in Cos7 cells assessed as luciferase activity after 24 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed