Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM50215716'
TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50215716(2-chloro-4-((3aS,4R)-4-hydroxy-3a-methyl-1,1,3-tri...)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]DHT from human androgen receptor in MDA453 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50215716(2-chloro-4-((3aS,4R)-4-hydroxy-3a-methyl-1,1,3-tri...)
Affinity DataEC50:  1.25E+3nMAssay Description:Agonist activity at androgen receptor in mouse C2C12 cells by receptor transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed