Affinity DataKi: 6nMAssay Description:Binding affinity to bicalutamide-resistant Androgen receptor T878A mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity to wild-type Androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Antagonist activity at wild type human recombinant androgen receptor assessed as inhibition of testosterone-induced growth of mouse androgen dependen...More data for this Ligand-Target Pair