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Found 3 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM50415098'
TargetAndrogen receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50415098(CHEMBL570898)
Affinity DataIC50:  2.5nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50415098(CHEMBL570898)
Affinity DataEC50:  15.8nMAssay Description:Agonist activity at androgen receptor in mouse NIH3T3 cells transiently transfected with beta-galactosidase reporter gene assessed as cellular transf...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50415098(CHEMBL570898)
Affinity DataEC50:  2.5nMAssay Description:Modulation of androgen receptor (unknown origin) expressed in Cos7 cells assessed as luciferase activity after 24 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed