Affinity DataIC50: 1.11E+3nMAssay Description:Antagonist activity at DHT-induced Androgen receptor transcriptional activity in human HEK293 cells measured after 24 hrs by Steady-Glo reagent based...More data for this Ligand-Target Pair
Affinity DataEC50: 405nMAssay Description:Displacement of [3H]R1881 from androgen receptor in human PC3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.04E+4nMAssay Description:Induction of degradation of full length Androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 845nMAssay Description:Displacement of [3H]R1881 from androgen receptor in human LNCAP cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 670nMAssay Description:Displacement of [3H]R1881 from AR in human LNCaP cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair