Affinity DataKi: 14nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Antagonist activity at Androgen receptor in human MDA-MB-453 cells measured by SEAP reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 125nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells measured by SEAP reporter gene assayMore data for this Ligand-Target Pair