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Found 2 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM93830'
TargetAndrogen receptor(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM93830(4-phenyl-2-(4-pyridyl)thiazole | 4-phenyl-2-pyridi...)
Affinity DataIC50:  630nMAssay Description:Inhibition of androgen receptor in human LNCaP cells assessed as inhibition of prostate-specific antigen secretion into media after 3 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM93830(4-phenyl-2-(4-pyridyl)thiazole | 4-phenyl-2-pyridi...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of androgen receptor transcriptional activity in human LNCaP cells after 3 days by eGFP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed