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Found 2 Enz. Inhib. hit(s) with Target = 'Angiopoietin-1 receptor' and Ligand = 'BDBM17789'
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Gsk

LigandPNGBDBM17789(benzimidazole-urea, 17 | methyl N-{6-[4-({[2-fluor...)
Affinity DataIC50:  6.90nMpH: 7.4 T: 2°CAssay Description:The assay uses purified GST-Tie-2 or GST-VEGFR2 interacting with biotinylated peptide substrates. HTRF is based on the proximity of europium cryptate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Gsk

LigandPNGBDBM17789(benzimidazole-urea, 17 | methyl N-{6-[4-({[2-fluor...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Tie2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed