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Found 2 Enz. Inhib. hit(s) with Target = 'Angiopoietin-1 receptor' and Ligand = 'BDBM50363397'
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50363397(CHEMBL1946170 | REGORAFENIB | US10183928, Regorafe...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of GST-tagged TIE2 (unknown origin) using biotin-Ahx-EPKDDAYPLYSDFG peptide as substrate by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAngiopoietin-1 receptor(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50363397(CHEMBL1946170 | REGORAFENIB | US10183928, Regorafe...)
Affinity DataIC50:  311nMAssay Description:Inhibition of Tie-2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank