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Found 5 Enz. Inhib. hit(s) with Target = 'Anoctamin-1' and Ligand = 'BDBM509678'
TargetAnoctamin-1(Homo sapiens (Human))
Enterprise Therapeutics

US Patent
LigandPNGBDBM509678(4-[[2-(2-Chlorophenyl)acetyl]amino]-N-(1-cyanocycl...)
Affinity DataEC50:  1.22E+3nMAssay Description:Compound activity was quantified by measuring the increase in current upon compound addition and expressing this as a percentage increase of baseline...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAnoctamin-1(Homo sapiens (Human))
Enterprise Therapeutics

US Patent
LigandPNGBDBM509678(4-[[2-(2-Chlorophenyl)acetyl]amino]-N-(1-cyanocycl...)
Affinity DataEC50:  220nMAssay Description:Compound activity was quantified by measuring the increase in current upon compound addition and expressing this as a percentage increase of baseline...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAnoctamin-1(Homo sapiens (Human))
Enterprise Therapeutics

US Patent
LigandPNGBDBM509678(4-[[2-(2-Chlorophenyl)acetyl]amino]-N-(1-cyanocycl...)
Affinity DataEC50:  220nMAssay Description:Cell Culture and PreparationFisher rat thyroid (FRT) cells stably expressing human TMEM16A (TMEM16Aabc variant; Dr Luis Galietta, Insituto Giannina, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAnoctamin-1(Homo sapiens (Human))
Enterprise Therapeutics

US Patent
LigandPNGBDBM509678(4-[[2-(2-Chlorophenyl)acetyl]amino]-N-(1-cyanocycl...)
Affinity DataEC50:  1.22E+3nMAssay Description:Cell Culture and PreparationFisher rat thyroid (FRT) cells stably expressing human TMEM16A (TMEM16Aabc variant; Dr Luis Galietta, Insituto Giannina, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAnoctamin-1(Homo sapiens (Human))
Enterprise Therapeutics

US Patent
LigandPNGBDBM509678(4-[[2-(2-Chlorophenyl)acetyl]amino]-N-(1-cyanocycl...)
Affinity DataEC50:  380nMAssay Description:Compound activity was quantified by measuring the increase in current upon compound addition and expressing this as a percentage increase of baseline...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent