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Found 6 Enz. Inhib. hit(s) with Target = 'Apelin receptor' and Ligand = 'BDBM270098'
TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM270098((1R,2S,P)—N-(4-(2-ethoxy-6-methoxyphenyl)-5-(...)
Affinity DataEC50:  0.310nMpH: 7.5Assay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV¿-3 expression vector (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM270098((1R,2S,P)—N-(4-(2-ethoxy-6-methoxyphenyl)-5-(...)
Affinity DataEC50:  3.90nMpH: 7.5Assay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV¿-3 expression vector (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM270098((1R,2S,P)—N-(4-(2-ethoxy-6-methoxyphenyl)-5-(...)
Affinity DataEC50:  3.90nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM270098((1R,2S,P)—N-(4-(2-ethoxy-6-methoxyphenyl)-5-(...)
Affinity DataEC50:  3.90nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM270098((1R,2S,P)—N-(4-(2-ethoxy-6-methoxyphenyl)-5-(...)
Affinity DataEC50:  0.310nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM270098((1R,2S,P)—N-(4-(2-ethoxy-6-methoxyphenyl)-5-(...)
Affinity DataEC50:  0.310nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent